GSK 525762A-d5

Chemical Name:GSK 525762A-d5
Synonyms:(4S)-6-(4-Chlorophenyl)-N-ethyl-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine-4-acetamide-d5; I-BET 762-d5;
Alternate CAS #:Unlabelled: 1260907-17-2
Molecular Formula:C₂₂H₁₇D₅ClN₅O₂
Molecular Weight:428.93
Category:Standards; Isotopic Labeled Analogues; Pharmaceutical/API Drug Impurities/Metabolites;
Applications:GSK 525762A-d5, is the labeled analogue of GSK 525762A (G797505), which is a BET Bromodomain Inhibitor currently in clinical development. BET bromodomains have emerged as promising drug targets for treatment of cancers, inflammatory diseases, and other medical conditions.
References:Zhao, Y., et al.: J. Med. Chem., 56, 7498 (2013); Mirguet, O., et al.: J. Med. Chem., 56, 7501 (2013);
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