CAS:130332-27-3|CI-988

Catalogue Number:C432695
Chemical Name:CI-988
Synonyms:4,9-Dihydro-4-[1-(methyl-d3)-4-piperidinylidene]-10H-benzo[4,5]cyclohepta[1,2-b]thiophen-10-one (2E)-2-Butenedioate; Ketotifen-d3 Hydrogen Fumarate; Totifen-d3; Zaditen-d3; Zaditor-d3; Zasten-d3;
CAS Number:130332-27-3
Molecular Formula:C23H20D3NO5S
Molecular Weight:614.73
Category:Research Tools;
Applications:CI-988 is a potent and selective cholecystokinin 2 (CCK-2) receptor antagonist that displays ~ 1600-fold selectivity over CCK1 receptors and has negligible affinity at other binding sites. CI-988 exhibits anxiolytic activity following oral administration. CI-98 inhibited the proliferation of small cell lung cancer (SCLC) cells in mice.
References:Drysdale, M. et al.: Bioorg. Med. Chem. Lett., 2, 45 (1992); Moody, T.W. et al.: J. Pharmacol. Exp. Ther., 299, 1154 (2001);
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