CAS:102146-07-6|8-Cyclopentyl-1,3-dipropylxanthine

Catalogue Number:C988500
Chemical Name:8-Cyclopentyl-1,3-dipropylxanthine
Synonyms:8-Cyclopentyl-3,9-dihydro-1,3-dipropyl-1H-purine-2,6-dione; DPCPX, PD 116,948
CAS Number:102146-07-6
Molecular Formula:C₁₆H₂₄N₄O₂
Appearance:White to Off-White Solid
Melting Point:194 – 197°C
Molecular Weight:304.39
Storage:-20°C
Solubility:Chloroform (Sparingly), Ethyl Acetate (Slightly, Heated, Sonicated), Methanol (S
Category:Standards; Enzyme Activators and Inhibitors; Neurochemicals;
Applications:DPCPX is a potent and very selective A1-adenosine receptor antagonist, with a Ki of 0.46 nM for A1 receptors in rat whole-brain membranes. Its 740-fold A1-selectivity is the highest reported for an adenosine antagonist.
References:Gessi, S., et al.: Mol. Pharmacol., 67, 2137 (2005), Minor, T.R., et al.: Behav. Neurosci., 122, 1236 (2008), Gracia, E., et al.: J. Neurochem., 107, 161 (2008), Gessi, S., et al.: Biochem. Pharmacol., 75, 562 (2008),
To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the products will be shipped in the box with layers of tapes to protect them against damage. The extremely low temperature products will be wrapped with dried ice, and the low temperature products will be delivered with ice bags. As for the products stored at room temperature, they will not be packed with ice bags or dried ice. Taskcm is committed to providing cost-effective products that facilitate drug delivery with our customers.
Email:sales@ebclink.com