Drug Delivery

Chemical Name:3-cis-HydroxyglipizideSynonyms:Hydroxycyclohexyl]amino]carbonyl]amino]sulfonyl]phenyl]ethyl]-5-methyl-2-pyrazinecarboxamide; 1-[4-[2-(5-Methylpyrazine-2-carboxamido)ethyl]phenylsulfonyl]-3-(3-cis-hydroxycyclohexyl)urea; N-[4-[β-(5-Methylpyrazine-2-carboxamido)ethyl]benzenesulfonyl]-N’-(3-cis-hydroxycyclohexyl)urea;CAS Number:38207-37-3Molecular Formula:C₂₁H₂₇N₅O₅SMolecular Weight:461.53Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:3-cis-Hydroxyglipizide is a metabolite of Glipizide (G410225), a sulfonylurea hypoglycemic agent. Used as an antidiabetic.References:Ambrogi, et al.: Arzneimittel-Forsch., 21, 200 (1971), Fuccella, et al.: J. Clin. Pharmacol., 13, 68 (1973), Brogden, R.N., et al.: Drugs, 18, 329 (1979), Lebovitz, H.E., et al.: Pharmacother., 5, 63 (1985)To […]

Chemical Name:7α-HydroxygliclazideSynonyms:rel-(3aα,5β,6aα)-N-[[(Hexahydrocyclopenta[c]pyrrol-2(1H)-yl)amino]carbonyl]-4-methyl-benzenesulfonamide; Cyclopenta[c]pyrrole, benzenesulfonamide deriv.CAS Number:96896-07-0Molecular Formula:C₁₅H₂₁N₃O₄SMolecular Weight:339.41Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:7α-Hydroxygliclazide is a metabolite of Gliclazide (G409875) which is a a sulfonylurea hypoglycemic agent used as an antidiabetic.References:Duhault, J., et al.: Arzneimittel-Forsch., 22, 1686 (1972), Holmes, B., et al.: Drugs, 27, 301 (1984),To ensure the stability of our products, the efficient express delivery service will […]

Chemical Name:7β-HydroxygliclazideSynonyms:rel-(3aα,5α,6aα)-N-[[(Hexahydro-5-hydroxycyclopenta[c]pyrrol-2(1H)-yl)amino]carbonyl]-4-methyl-benzenesulfonamide; 5-Hydroxy-hexahydro-cyclopenta[c]pyrrole BenzenesulfonamideCAS Number:96860-48-9Molecular Formula:C₁₅H₂₁N₃O₄SMolecular Weight:339.41Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:7β-Hydroxygliclazide is a metabolite of Gliclazide (G409875) which is a a sulfonylurea hypoglycemic agent used as an antidiabetic.References:Duhault, J., et al.: Arzneimittel-Forsch., 22, 1686 (1972), Holmes, B., et al.: Drugs, 27, 301 (1984),To ensure the stability of our products, the efficient express delivery service will be […]

Chemical Name:Hydroxy Famciclovir-d4Alternate CAS #:unlabelled: 172645-79-3Molecular Formula:C₁₄H₁₅D₄N₅O₅Molecular Weight:341.36Category:Standards; Isotopic Labeled Analogues;Applications:Hydroxy Famciclovir-d4 is the labelled analogue of Hydroxy Famciclovir, which is a Famciclovir (F101125) derivative and may be a useful hepadnaviridae-active antiviral agent.References:Marcuccio, S. M., et al.: PCT Int. Appl. WO 9522330 A1 19950824 (1995)To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that […]

Chemical Name:5-Hydroxyfraxetin 8-beta-D-GlucosideSynonyms:5,7-Dihydroxy-6-methoxy-8-(((2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)oxy)-2H-chromen-2-one; 5,7-Dihydroxy-6-methoxycoumarin 8-β-D-Glucoside; 5,7-Dihydroxy-6-methoxycoumarin 8-β-D-GlucopyranosideMolecular Formula:C₁₆H₁₈O₁₁Molecular Weight:386.31Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites; Carbohydrates and Oligosaccharides;Applications:5-Hydroxyfraxetin 8-β-D-Glucoside is a derivative of Fraxetin (F763960); a coumarin compound with anti-oxidant and anti-inflammatory activity. It also acts as a protective agent against hyperuricemia and renal dysfunction.References:Witaicenis, A. et al.: Phytomed. 21, 240 (2014); Chen, X. et al.: Int. Immunopharm., […]

Chemical Name:6’-Hydroxy N-Desisopropyl Delavirdine-d8Synonyms:N-[2-[[4-(3-Amino-1,6-dihydro-6-oxo-2-pyridinyl)-1-piperazinyl]carbonyl]-1H-indol-5-yl]methanesulfonamide-d8; 1-(3-Amino-1,6-dihydro-6-oxo-2-pyridinyl)-4-[[5-[(methylsulfonyl)amino]-1H-indol-2-yl]carbonyl]piperazine-d8Alternate CAS #:Unlabelled: 188780-41-8Molecular Formula:C₁₉H₁₄D₈N₆O₄SMolecular Weight:438.53Category:Standards; Isotopic Labeled Analogues; Pharmaceutical/API Drug Impurities/Metabolites;Applications:6’-Hydroxy N-Desisopropyl Delavirdine-d8 is the isotope labelled analog of 6’-Hydroxy N-Desisopropyl Delavirdine (H936540); a metabolite of Delavirdine (D230625) which is a bisheteroarylpiperazine (BHAP) reverse transcriptase inhibitor.References:Dueweke, T.J., et al.: Antimicrob. Ag. Chemother., 37, 1127 (1993); Althaus, I.W., et al.: Biochem. […]

Chemical Name:6’-Hydroxy N-Desisopropyl DelavirdineSynonyms:N-[2-[[4-(3-Amino-1,6-dihydro-6-oxo-2-pyridinyl)-1-piperazinyl]carbonyl]-1H-indol-5-yl]methanesulfonamide; 1-(3-Amino-1,6-dihydro-6-oxo-2-pyridinyl)-4-[[5-[(methylsulfonyl)amino]-1H-indol-2-yl]carbonyl]piperazineCAS Number:188780-41-8Molecular Formula:C₁₉H₂₂N₆O₄SMolecular Weight:430.48Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:6’-Hydroxy N-Desisopropyl Delavirdine is a metabolite of Delavirdine (D230625); a bisheteroarylpiperazine (BHAP) reverse transcriptase inhibitor.References:Dueweke, T.J., et al.: Antimicrob. Ag. Chemother., 37, 1127 (1993); Althaus, I.W., et al.: Biochem. Pharmacol., 47, 2017 (1994); Chang, M., et al.: Drug Metab. Dispos., 25, 228 (1997)To ensure the […]

Chemical Name:1β-Hydroxydeoxycholic Acid-d4 (major)Synonyms:(1β,​3α,​5β,​12α)​-1,​3,​12-​Trihydroxy-​cholan-​24-​oic-​2,​2,​4,​4-​d4 AcidCAS Number:2089602-33-3Alternate CAS #:Unlabelled: 80434-32-8Molecular Formula:C₂₄H₃₆D₄O₅Molecular Weight:412.6Category:Standards; Isotopic Labeled Analogues; Pharmaceutical/API Drug Impurities/Metabolites; Steroids;Applications:1β-Hydroxydeoxycholic Acid-d4 is the isotope labelled analog of 1β-Hydroxydeoxycholic Acid (H934880); a metabolite of Taurodeoxycholic Acid (T009000) which is a steroidal amphipathic hepatic bile salt formed in the liver through the conjugation of Deoxycholate (S624090) with Taurine (T007850).References:Gutasfsson, […]

Chemical Name:1beta-Hydroxydeoxycholic AcidSynonyms:1β,3α,12α-Trihydroxy-5β-cholan-24-oic Acid; 1β,3α,12α-Trihydroxy-5β-cholanoic Acid; (1β,3α,5β,12α)-1,3,12-Trihydroxycholan-24-oic Acid;CAS Number:80434-32-8Molecular Formula:C₂₄H₄₀O₅Molecular Weight:408.57Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites; Steroids;Applications:1β-Hydroxydeoxycholic Acid is an metabolite of Taurodeoxychloic Acid (T009000), a steroidal amphipathic hepatic bile salt formed in the liver through the conjugation of deoxycholate (S624090) with taurine (T007850).References:Gutasfsson, J., et al.: Biol. Neonate., 47, 26 (1985); Shoda, J., et al.: J. […]

Chemical Name:6’-Hydroxy Delavirdine-d8Synonyms:N-[2-[[4-[1,6-Dihydro-3-[(1-methylethyl)amino]-6-oxo-2-pyridinyl]-1-piperazinyl]carbonyl]-1H-indol-5-yl]methanesulfonamide-d8; 1-[1,6-Dihydro-3-[(1-methylethyl)amino]-6-oxo-2-pyridinyl]-4-[[5-[(methylsulfonyl)amino]-1H-indol-2-yl]carbonyl]piperazine-d8Alternate CAS #:Unlabelled: 188780-44-1Molecular Formula:C₂₂H₂₀D₈N₆O₄SMolecular Weight:480.61Category:Standards; Isotopic Labeled Analogues; Pharmaceutical/API Drug Impurities/Metabolites;Applications:6’-Hydroxy Delavirdine-d8 is the isotope labelled analog of 6’-Hydroxy Delavirdine (H934505); a metabolite of Delavirdine (D230625) which is a bisheteroarylpiperazine (BHAP) reverse transcriptase inhibitor.References:Dueweke, T.J., et al.: Antimicrob. Ag. Chemother., 37, 1127 (1993); Althaus, I.W., et al.: Biochem. Pharmacol., 47, 2017 […]