Drug Delivery

Chemical Name:6’-Hydroxy DelavirdineSynonyms:N-[2-[[4-[1,6-Dihydro-3-[(1-methylethyl)amino]-6-oxo-2-pyridinyl]-1-piperazinyl]carbonyl]-1H-indol-5-yl]methanesulfonamide; 1-[1,6-Dihydro-3-[(1-methylethyl)amino]-6-oxo-2-pyridinyl]-4-[[5-[(methylsulfonyl)amino]-1H-indol-2-yl]carbonyl]piperazineCAS Number:188780-44-1Molecular Formula:C₂₂H₂₈N₆O₄SMolecular Weight:472.56Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:6’-Hydroxy Delavirdine is a metabolite of Delavirdine (D230625); a bisheteroarylpiperazine (BHAP) reverse transcriptase inhibitor.References:Dueweke, T.J., et al.: Antimicrob. Ag. Chemother., 37, 1127 (1993); Althaus, I.W., et al.: Biochem. Pharmacol., 47, 2017 (1994); Voorman, R.L., et al.: J. Pharmacol. Exp. Ther., 287, 381 (1998)To ensure the stability […]

Chemical Name:3-Hydroxy Cyclobenzaprine-d6Synonyms:5-[3-(Dimethylamino)propylidene]-5H-dibenzo[a,d]cyclohepten-3-ol-d6;CAS Number:1217246-95-1Alternate CAS #:unlabelled: 30235-48-4Molecular Formula:C₂₀H₁₅D₆NOMolecular Weight:297.42Category:Standards; Isotopic Labeled Analogues; Pharmaceutical/API Drug Impurities/Metabolites;Applications:A labelled metabolite of Cyclobenzaprine (C987750).References:Hucker, H.B., et al.: Drug Metab. Dispos., 6, 184-92 (1978),To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the products will be shipped in the box […]

Chemical Name:3,16-Dihydroxycorticosterone 20-Hydroxy-21-AcidMolecular Formula:C₂₁H₃₂O₆Molecular Weight:380.48Category:Standards; Chiral Molecules; Pharmaceutical/API Drug Impurities/Metabolites; Steroids;Applications:3,16-Dihydroxycorticosterone 20-Hydroxy-21-Acid is a derivative of Corticosterone (C695700), an intermediate in the biosynthesis of Aldosterone (A514700), isolated from the adrenal cortex.References:Schmidt, M., et al.: Endocrinol., 150, 2709 (2009), Bailey, M., et al.: J. Immunol., 182, 7888 (2009), Brunton, P., et al.: J. Neurosci., 29, 6449 […]

Chemical Name:6-​β-​Hydroxycortisol-d4 SulfateSynonyms:6-β-Hydroxycortisol-d4 MonosulfateAlternate CAS #:Unlabelled: 53587-06-7Molecular Formula:C₂₁H₂₆D₄O₉SMolecular Weight:462.55Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites; Steroids;Applications:Isotope labelled 6-β-Hydroxycortisol Sulfate is used in the synthesis of corticosteroids in human blood.References:Miyabo, S. et al.: J. Steroid. Biochem., 5, 233 (1974);To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the products […]

Chemical Name:24-Hydroxy Cabotegravir-d3Synonyms:(3S,11aR)-N-(2,4-Difluoro-3-hydroxybenzyl)-6-hydroxy-3-methyl-5,7-dioxo-2,3,5,7,11,11a-hexahydrooxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamide-d3Molecular Formula:C₁₉H₁₄D₃F₂N₃O₆Molecular Weight:424.37Category:Standards; Isotopic Labeled Analogues; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;Applications:24-Hydroxy Cabotegravir-d3 is the labelled form of 24-Hydroxy Cabotegravir. 24-Hydroxy Cabotegravir is a metabolite of Cabotegravir (C050100). Cabotegravir is a long acting HIV-1 integrase inhibitor with action against a broad range of HIV subtypes.References:Yoshinaga, T. et al.: Antimicrob, Agents Chemother., 59, […]

Chemical Name:24-Hydroxy CabotegravirSynonyms:(3S,11aR)-N-(2,4-Difluoro-3-hydroxybenzyl)-6-hydroxy-3-methyl-5,7-dioxo-2,3,5,7,11,11a-hexahydrooxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamideMolecular Formula:C₁₉H₁₇F₂N₃O₆Molecular Weight:421.35Category:Standards; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;Applications:24-Hydroxy Cabotegravir is a metabolite of Cabotegravir (C050100). Cabotegravir is a long acting HIV-1 integrase inhibitor with action against a broad range of HIV subtypes.References:Yoshinaga, T. et al.: Antimicrob, Agents Chemother., 59, 397 (2015); Andrews, C. et al.: Sci. Transl. Med., 7, 270 (2015)To […]

Chemical Name:13-Hydroxy Cabotegravir-d3Synonyms:(3S,11aR)-N-(2,4-Difluorobenzyl)-2,6-dihydroxy-3-methyl-5,7-dioxo-2,3,5,7,11,11a-hexahydrooxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamide-d3Molecular Formula:C₁₉H₁₄D₃F₂N₃O₆Molecular Weight:424.37Category:Standards; Isotopic Labeled Analogues; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;Applications:13-Hydroxy Cabotegravir-d3 is the labelled form of 13-Hydroxy Cabotegravir. 13-Hydroxy Cabotegravir is a metabolite of Cabotegravir (C050100). Cabotegravir is a long acting HIV-1 integrase inhibitor with action against a broad range of HIV subtypes.References:Yoshinaga, T. et al.: Antimicrob, Agents Chemother., 59, […]

Chemical Name:13-Hydroxy CabotegravirSynonyms:(3S,11aR)-N-(2,4-Difluorobenzyl)-2,6-dihydroxy-3-methyl-5,7-dioxo-2,3,5,7,11,11a-hexahydrooxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamideMolecular Formula:C₁₉H₁₇F₂N₃O₆Molecular Weight:421.35Category:Standards; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;Applications:13-Hydroxy Cabotegravir is a metabolite of Cabotegravir (C050100). Cabotegravir is a long acting HIV-1 integrase inhibitor with action against a broad range of HIV subtypes.References:Yoshinaga, T. et al.: Antimicrob, Agents Chemother., 59, 397 (2015); Andrews, C. et al.: Sci. Transl. Med., 7, 270 (2015)To […]

Chemical Name:4-Hydroxycarbazeran-d4Synonyms:1-(3,4-Dihydro-6,7-dimethoxy-4-oxo-1-phthalazinyl)-4-piperidinyl Ester Ethylcarbamic Acid-d4;Alternate CAS #:Unlabelled: 96724-43-5Molecular Formula:C₁₈H₂₀D₄N₄O₅Molecular Weight:380.43Category:Building Blocks; Isotopic Labeled Analogues;Applications:4-Hydroxycarbazeran-d4 is the isotope labelled analog of 4-Hydroxycarbazeran, a metabolite of Carbazeran (C175790). Carbazeran is known as a phosphodiesterase inhibitor drug that exhibits chronictropic and inotropic effects.References:Kaye, B., et al.: Xenobiotica., 15, 237 (1985); Shahid, M., et al.: Br. J. Pharmacol., 98, 291 […]

Chemical Name:4-Hydroxy Atorvastatin Acyl-β-D-glucuronide 80%, contains up to 20% lactoneSynonyms:(βR,δR)-2-(4-Fluorophenyl)-β,δ-dihydroxy-4-[[(4-hydroxyphenyl)amino]carbonyl]-5-(1-methylethyl)-3-phenyl-1H-pyrrole-1-heptanoic Acid β-D-Glucopyranuronic Acid;Molecular Formula:C₃₉H₄₃FN₂O₁₂Molecular Weight:750.76Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:A metabolite of Atorvastatin (A791750).To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the products will be shipped in the box with layers of tapes to protect them […]